Generic (Common) Name | Brand Name | Company | Year Approved |
Protease Inhibitors (PIs) | |||
amprenavir | Agenerase | GlaxoSmithKline | 1999; withdrawn 2007 |
atazanavir | Reyataz | Bristol-Myers Squibb | 2003 |
darunavir | Prezista | Tibotec | 2006 |
fosamprenavir | Lexiva (U.S.) Telzir (Europe) | ViiV Healthcare | 2003 |
indinavir | Crixivan | Merck | 1996 |
lopinavir/ritonavir | Kaletra | Abbott | 2000; Meltrex formulation 2005 |
nelfinavir | Viracept | ViiV Healthcare | 1997 |
ritonavir | Norvir | Abbott | 1996 |
saquinavir | Invirase (hard gel) Fortovase (soft gel) | Roche | 1995 1997; withdrawn 2005 |
tipranavir | Aptivus | Boehringer Ingelheim | 2005 |
Nucleoside/Nucleotide Reverse Transcriptase Inhibitors (NRTIs) | |||
abacavir | Ziagen | ViiV Healthcare | 1998 |
didanosine (ddI) | Videx | Bristol-Myers Squibb | 1989; Videx EC 2000 |
emtricitabine (FTC) | Emtriva | Gilead | 2003 |
lamivudine (3TC) | Epivir | ViiV Healthcare | 1995 |
stavudine (d4T) | Zerit | Bristol-Myers Squibb | 1994 |
tenofovir DF | Viread | Gilead | 2002 |
zalcitabine (ddC) | Hivid | Roche | 1992; withdrawn 2005 |
zidovudine (AZT) | Retrovir | ViiV Healthcare | 1987 |
Non-Nucleoside Reverse Transcriptase Inhibitors (NNRTIs) | |||
delavirdine | Rescriptor | ViiV Healthcare | 1997 |
efavirenz | Sustiva (U.S.) Stocrin (elsewhere) | Bristol-Myers Squibb | 1998 |
etravirine | Intelence | Tibotec | 2008 |
nevirapine | Viramune | Boehringer Ingelheim | 1996 |
Other Classes | |||
enfuvirtide (T-20; fusion inhibitor) | Fuzeon | Roche/Trimeris | 2003 |
maraviroc (CCR5 antagonist) | Selzentry (U.S.) Celsentri (elsewhere) | ViiV Healthcare | 2007 |
raltegravir (integrase inhibitor) | Isentress | Merck | 2007 |
Fixed-Dose Combinations | |||
lamivudine/abacavir (NRTI) | Epzicom (U.S.) Kivexa (Europe) | ViiV Healthcare | 2004 |
tenofovir/emtricitabine (NRTI) | Truvada | Gilead | 2004 |
tenofovir/emtricitabine/efavirenz (NRTI/NNRTI) | Atripla | Gilead/Bristol-Myers Squibb | 2006 |
zidovudine/lamivudine (NRTI) | Combivir | ViiV Healthcare | 1997 |
zidovudine/lamivudine/abacavir (NRTI) | Trizivir | ViiV Healthcare | 2000 |
This article was originally published January 1, 2010 and most recently updated March 1, 2010.
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